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Product Description
– BET bromodomain inhibitor 2 is a potent BET bromodomain inhibitor with an IC50 of 14.1 µM[1].
Web ID
– HY-146709
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C23H30N2O5S
References
– [1]J P Hilton-Proctor, et al. Substituted 1-methyl-4-phenylpyrrolidin-2-ones – Fragment-based design of N-methylpyrrolidone-derived bromodomain inhibitors. Eur J Med Chem. 2020 Apr 1;191:112120.
CAS Number
– 2414195-69-8
Molecular Weight
– 446.56
SMILES
– CCN(S(=O)(C1=CC=C(C(C2=CC(OC)=C(C=C2)OC)=C1)[C@H]3CC(N(C3)C)=O)=O)CC
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
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