Download Files:
Azatadine (dimaleate)
$38 – $180
Products Details
Product Description
– Azatadine bimaleate is an inhibitor of histamine receptors and choline receptors with IC50s of 6.5 nM and 10 nM respectively.
Web ID
– HY-B0170A
Storage Temperature
– 4°C (Powder, sealed storage, away from moisture)
Shipping
– Room Temperature
Applications
– COVID-19-immunoregulation
Molecular Formula
– C28H30N2O8
References
– [1]Wilson JD, et al. Azatadine maleate (Zadine): evaluation in the management of allergic rhinitis. N Z Med J. 1981 Aug 12;94(689):79-81.|[2]Tozzi S, et al. The pharmacology of azatadine, a potential antiallergy drug. Agents Actions. 1974 Oct;4(4):264-70.
CAS Number
– 3978-86-7
Molecular Weight
– 522.55
Compound Purity
– 99.85
SMILES
– O=C(O)/C=CC(O)=O.O=C(O)/C=CC(O)=O.CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=CC=CN=C42
Clinical Information
– Launched
Research Area
– Inflammation/Immunology; Endocrinology
Solubility
– DMSO : ≥ 100 mg/mL|H2O : ≥ 100 mg/mL
Target
– Histamine Receptor
Pathway
– GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
