Atipamezole

$61$312

Products Details

Product Description

– Atipamezole (MPV 1248) is a potent α2-adrenoceptor antagonist with a Ki of 1.6 nM[1].

Web ID

– HY-12380A

Storage Temperature

– -20°C, 3 years; 4°C, 2 years (Powder)

Shipping

– Room Temperature

Applications

– Neuroscience-Neuromodulation

Molecular Formula

– C14H16N2

Citations

– Brain Res. 2020 Sep 15;1743:146949.|Eur J Neurosci. 2021 Apr 27.|Exp Mol Pathol. 2021 Feb;118:104587.|Front Cell Dev Biol. 2021 Mar 11;9:636327.|Research Square Preprint. 2022 May.|Sci Transl Med. 2022 Nov 3;eabq4064.|Protein Cell. 2019 Mar;10(3):178-195.

References

– [1]Pertovaara A, et al.Pharmacological properties, central nervous system effects, and potential therapeutic applicationsof atipamezole, a selective alpha2-adrenoceptor antagonist. CNS Drug Rev. 2005 Autumn;11(3):273-88.

CAS Number

– 104054-27-5

Molecular Weight

– 212.29

Compound Purity

– 99.74

SMILES

– CCC1(C2=CN=CN2)CC3=C(C=CC=C3)C1

Clinical Information

– Phase 1

Research Area

– Neurological Disease; Endocrinology

Solubility

– DMSO : ≥ 30 mg/mL

Target

– Adrenergic Receptor

Isoform

– α adrenergic receptor

Pathway

– GPCR/G Protein;Neuronal Signaling

Product type

– Reference compound

Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.

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