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AR antagonist 2
SKU
HY-142923-Get quote
Category Reference compound
Tags Androgen Receptor, Cancer, Vitamin D Related/Nuclear Receptor
Products Details
Product Description
– AR antagonist 2 (compound 58) is a potent androgen receptor (AR) inhibitor with an IC50 of 0.95 μM. AR antagonist 2 has the potential for cancer research[1].
Web ID
– HY-142923
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C22H17ClFN5O2S
References
– [1]Chenli Shen, et al. Diaryl thiohydantoins as androgen receptor antagonists. WO2019029521A1
CAS Number
– 2275752-15-1
Molecular Weight
– 469.92
SMILES
– N#CC1=CC=C(N(C(N(C2=CN(C(C(F)=C2)=NC(CC)=C3)C3=O)C4(C)C)=S)C4=O)C=C1Cl
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Androgen Receptor
Pathway
– Vitamin D Related/Nuclear Receptor
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.