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ALDH1A2-IN-1
$170 – $1,280
Products Details
Product Description
– ALDH1A2-IN-1 is an active site-directed reversible ALDH1A2 inhibitor (IC50=0.91 μM; Kd=0.26 μM) with several hydrophobic interactions[1].
Web ID
– HY-139031
Storage Temperature
– -20°C, 3 years (Powder)
Shipping
– Blue Ice
Applications
– Metabolism-sugar/lipid metabolism
Molecular Formula
– C21H26N4O4S
References
– [1]Chen Y, et al. Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors. ACS Chem Biol. 2018;13(3):582-590.
CAS Number
– 2204229-64-9
Molecular Weight
– 430.52
Compound Purity
– 98.80
SMILES
– O=C(C1=C(OCC)C=CS1)N2CCN(C3=CC=C([N+]([O-])=O)C(N4CCCC4)=C3)CC2
Clinical Information
– No Development Reported
Research Area
– Endocrinology
Solubility
– DMSO : 25 mg/mL (ultrasonic;warming;heat to 60°C)
Target
– Aldehyde Dehydrogenase (ALDH)
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
