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A2B receptor antagonist 2
SKU
HY-139314-100 mg
Category Reference compound
Tags Adenosine Receptor, GPCR/G Protein, Metabolic Disease
$60 – $140
Products Details
Product Description
– A2B receptor antagonist 2 (compound 18) is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively[1].
Web ID
– HY-139314
Storage Temperature
– 4°C (Powder, protect from light)
Shipping
– Room Temperature
Applications
– Metabolism-protein/nucleotide metabolism
Molecular Formula
– C12H15N5
References
– [1]Thomas R Webb, et al. Quinazolines as adenosine receptor antagonists: SAR and selectivity for A2B receptors. Bioorg Med Chem. 2003 Jan 2;11(1):77-85.
CAS Number
– 784-90-7
Molecular Weight
– 229.28
Compound Purity
– 99.88
SMILES
– NC(NC1=NC(C)=C2C=C(C)C(C)=CC2=N1)=N
Clinical Information
– No Development Reported
Research Area
– Metabolic Disease
Solubility
– DMSO : 2 mg/mL (ultrasonic;warming;heat to 60°C)
Target
– Adenosine Receptor
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.