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Products Details
Product Description
– A-123189 is a selective and potent α1D antagonist with Kis of 0.312 and 0.17 for human α1D and rat α1D, respectively. A-123189 displays selectivities between 10- to 20-fold for the α1D receptor over the human α1A and rat α1A receptors[1].
Web ID
– HY-116623
Shipping
– Room temperature
Molecular Formula
– C26H28N4O3S
References
– [1]K P Briski, et al. Antagonism of type II, but not type I glucocorticoid receptors results in elevated basal luteinizing hormone release in male rats. Bioorganic & Medicinal Chemistry Letters, Volume 11, Issue 9, 7 May 2001, Pages 1119-1121.
CAS Number
– 255713-53-2
Molecular Weight
– 476.59
SMILES
– O=C1N(C(C2=C(N1)SC=C2C3=CC=CC(C)=C3)=O)CCN4CCN(CC4)C5=CC=CC=C5OC
Clinical Information
– No Development Reported
Research Area
– Endocrinology
Solubility
– 10 mM in DMSO
Target
– Adrenergic Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
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