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Products Details
Product Description
– 5-HT7R antagonist 1 is a G protein-biased antagonist against 5-HT7R (Ki = 6.5 nM).
Web ID
– HY-139677
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C14H18Cl2N4
References
– [1]Kwag R, et al. Discovery of G Protein-Biased Antagonists against 5-HT7R. J Med Chem. 2021 Sep 23;64(18):13766-13779.
CAS Number
– 2759919-13-4
Molecular Weight
– 313.23
SMILES
– ClC1=CC(C2=NNC=C2N3CCCNCC3)=CC=C1.Cl
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– G protein-coupled Bile Acid Receptor 1
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
