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Products Details
Product Description
– 5-HT7 receptor ligand 1 (Compound 5c) is a 5-HT7 receptor ligand with a Ki of 8 nM. 5-HT7 receptor ligand 1 is not hepatotoxic and exhibit moderate potential interaction with other agents metabolized by CYP3A4 or CYP2D6[1].
Web ID
– HY-147810
Shipping
– Room temperature
Applications
– Neuroscience-Neuromodulation
Molecular Formula
– C21H23N7
References
– [1]Kułaga D, et al. Aminotriazines with indole motif as novel, 5-HT7 receptor ligands with atypical binding mode. Bioorg Chem. 2020 Nov;104:104254.
CAS Number
– 2758571-64-9
Molecular Weight
– 373.45
SMILES
– NC1=NC(NCCC2=CNC3=C2C=CC=C3)=NC(NCCC4=CC=CC=C4)=N1
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– 5-HT Receptor
Isoform
– 5-HT7 Receptor
Pathway
– GPCR/G Protein;Neuronal Signaling
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
