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3-Hydroxyphenazepam
SKU
HY-124030-1mg
Category Reference compound
Tags Drug Metabolite, Metabolic Enzyme/Protease, Neurological Disease
$130
Only 1000 item(s) left in stock.
Products Details
Product Description
– 3-Hydroxyphenazepam is an active metabolite of Cinazepam. Cinazepam is a GABAA receptor agonist. 3-Hydroxyphenazepam can inhibit synaptosomal transporter-mediated [3H]GABA uptake[1].
Web ID
– HY-124030
Shipping
– Room temperature
Molecular Formula
– C15H10BrClN2O2
References
– [1]Borisova T, et, al. GABAA receptor agonist cinazepam and its active metabolite 3-hydroxyphenazepam act differently at the presynaptic site. Eur Neuropsychopharmacol. 2021 Apr;45:39-51.
CAS Number
– 70030-11-4
Molecular Weight
– 365.61
SMILES
– BrC1=CC(C(C2=CC=CC=C2Cl)=NC3O)=C(C=C1)NC3=O
Clinical Information
– No Development Reported
Research Area
– Neurological Disease
Solubility
– 10 mM in DMSO
Target
– Drug Metabolite
Pathway
– Metabolic Enzyme/Protease
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.