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Products Details
Product Description
– 2-(2,6-Dioxopiperidin-3-yl)phthalimidine-C5-Br is a E3 ligase ligand-linker conjugate for PROTAC.
Web ID
– HY-132939
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C18H21BrN2O3
References
– [1]Wei D, et al. Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer. J Med Chem. 2021 Oct 14;64(19):14822-14847.
CAS Number
– 2411022-24-5
Molecular Weight
– 393.27
SMILES
– O=C(C(N(CC1=C2C=CC=C1CCCCCBr)C2=O)CC3)NC3=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– E3 Ligase Ligand-Linker Conjugates
Pathway
– PROTAC
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
