Download Files:
(αR,8aS)-GSK1614343
$510 – $4,200
Products Details
Product Description
– (αR,8aS)-GSK1614343 (compound 18a, d2) is a cyclized ghrelin antagonist with an pIC50 value of 8.4. (αR,8aS)-GSK1614343 shows a competitive antagonism of hGHSR1a with a mean pKb value of 8.06[1].
Web ID
– HY-113906A
Storage Temperature
– -20°C, 3 years (Powder)
Shipping
– Blue Ice
Applications
– COVID-19-immunoregulation
Molecular Formula
– C22H23F6N5O
References
– [1]https://pubmed.ncbi.nlm.nih.gov/20593439/
CAS Number
– 1092476-84-0
Molecular Weight
– 487.44
Compound Purity
– 99.40
SMILES
– FC(F)(F)C1=CC(C(F)(F)F)=CC(NNC([C@@H](C2=CN=CC=C2)N3C[C@@]4([H])N(CCC4)CC3)=O)=C1
Clinical Information
– No Development Reported
Research Area
– Inflammation/Immunology
Solubility
– DMSO : 100 mg/mL (ultrasonic)
Target
– GHSR
Pathway
– GPCR/G Protein
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
