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Products Details
Product Description
– BRD4-BD1/2-IN-1 is a potent BRD4 inhibitor with IC50s of <100 nM for BRD4 BD-1 and BRD4 BD-2, respectively (US20150148375A1, compound 5)[1].
Web ID
– HY-142674
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C21H14F2N4O2
References
– [1]Bicyclic heterocycles as bet protein inhibitors. US20150148375A1.
CAS Number
– 1781219-19-9
Molecular Weight
– 392.36
SMILES
– O=C1C2=C(C(C3=CC4=C(C=C3OC5=CC=C(C=C5F)F)N=CN4)=CN1C)C=CN2
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
