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ARD-2585
$960 – $7,900
Products Details
Product Description
– ARD-2585 is an exceptionally potent and orally active PROTAC degrader of androgen receptor[1].
Web ID
– HY-139436
Storage Temperature
– -20°C (Powder, sealed storage, away from moisture and light)
Shipping
– Blue Ice
Applications
– Cancer-programmed cell death
Molecular Formula
– C41H43ClN8O5
References
– [1]Weiguo Xiang. et al. Discovery of ARD-2585 as an Exceptionally Potent and Orally Active PROTAC Degrader of Androgen Receptor for the Treatment of Advanced Prostate Cancer. J Med Chem. 2021 Sep 23;64(18):13487-13509.
CAS Number
– 2757422-79-8
Molecular Weight
– 763.28
Compound Purity
– 99.48
SMILES
– O=C(N(C1C(NC(CC1)=O)=O)C2=O)C(C2=C3)=CC=C3N(C4)CC4N(CC5)CCN5C(C=C6)=CC=C6C(N[C@@H]7CC[C@@H](N(C)C8=CC=C(C#N)C(Cl)=C8)CC7)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– DMSO : 85 mg/mL (ultrasonic)
Target
– Androgen Receptor;PROTACs
Pathway
– PROTAC;Vitamin D Related/Nuclear Receptor
Product type
– Reference compound
Disclaimer: All products are for research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation.
