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Products Details
Product Description
– GSK232 is a highly selective, cellularly penetrant CECR2 inhibitor with excellent physicochemical properties.
Web ID
– HY-145347
Shipping
– Room temperature
Applications
– Cancer-programmed cell death
Molecular Formula
– C21H27ClN6O3S
References
– [1]Lucas SCC, et al. Optimization of Potent ATAD2 and CECR2 Bromodomain Inhibitors with an Atypical Binding Mode. J Med Chem. 2020 May 28;63(10):5212-5241.
CAS Number
– 2702984-69-6
Molecular Weight
– 479.00
SMILES
– O=S(C(C=C1NC(CN2C3=C(CN(CC3)C)N=N2)=O)=C(C=C1)Cl)(N4C[C@@](C5CC5)([H])CC4)=O
Clinical Information
– No Development Reported
Research Area
– Cancer
Solubility
– 10 mM in DMSO
Target
– Epigenetic Reader Domain
Pathway
– Epigenetics
Product type
– Reference compound
Disclaimer: All products are for Research use only unless clearly stated otherwise on the product datasheet. Datasheets provided on the website are drafts for reference purpose only and you are requested to always refer to the hard copy included in the kit for your experimentation. Agdia Products are available for delivery only in Canada.
